阻害剤
タンパク質や酵素活性を遮断または低下させる化合物
化学原料を購入する必要がある場合は、 要求情報を送信してください最新の見積りを入手してください。
阻害剤の学術論文
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Novel inhibitors of the gardos channel for the treatment of sickle cell disease
関連化学物質
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Benzenemethanol, 2-fluoro-a-(4-fluorophenyl)-a-phenyl-
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Iodo and diiodotyrosine epoxysuccinyl derivatives as selective inhibitors of cathepsin B
関連化学物質
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パパイン
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L-trans-epoxysuccinyl-L-tyrosylamido(3-methyl)butane ethylester
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Discovery of
aSeries of Indole-2 Carboxamides as Selective Secreted Phospholipase A2 Type X (sPLA2-X) Inhibitors関連化学物質
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6-(trifluoromethoxy)-1H-indole-2-carboxylic acid
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Synthesis and biological evaluation of penam sulfones as inhibitors of β-lactamases
関連化学物質
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benzhydryl 2β-(chloroacetoxy)methyl-1,1-dioxo-penicillanate
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Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 1: Substitution of the glycine carboxylic acid group
関連化学物質
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Carbamic acid, [[1-(phenylmethyl)-1H-tetrazol-5-yl]methyl]-, 1,1-dimethylethyl ester
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Prostaglandin Synthetase Inhibitors from the African Medicinal Plant
関連化学物質
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Benzoic acid, 2-methoxy-6-(1-pentadecenyl)-, ethyl ester, (Z)-
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Synthesis and evaluation of inhibitors of bacterial drug efflux pumps of the major facilitator superfamily
関連化学物質
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2-NAPHTHYL ISOCYANIDE 97
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Inhibitors of Cholesterol Biosynthesis. 3. Tetrahydro-4-hydroxy-6-<2-(1H-pyrrol-1-yl)ethyl>-2H-pyran-2-one Inhibitors of HMG-CoA Reductase. 2. Effects of Introducing Substituents at Positions Three and Four of the Pyrrole Nucleus
関連化学物質
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dimethyl 1-<2-(1,3-dioxolan-2-yl)ethyl>-2-(4-fluorophenyl)-5-(1-methylethyl)-1H-pyrrole-3,4-dicarboxylate
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Discovery of a novel and potent series of dianilinopyrimidineurea and urea isostere inhibitors of VEGFR2 tyrosine kinase
関連化学物質
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Benzene, 1-[(methylsulfonyl)methyl]-3-nitro-
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Discovery of novel P-glycoprotein-mediated multidrug resistance inhibitors bearing triazole core via click chemistry
関連化学物質
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ジクロロメタン（別名塩化メチレン）
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トリエチルアミン
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N-(2-((1-(4-(2-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)phenyl)-1H-1,2,3-triazol-4-yl)methoxy)phenyl)benzamide
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The discovery and development of selective 3-fluoro-4-aryloxyallylamine inhibitors of the amine oxidase activity of semicarbazide-sensitive amine oxidase/vascular adhesion protein-1 (SSAO/VAP-1)
関連化学物質
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(E)-tert-butyl (4-hydroxybut-2-en-1-yl)carbamate
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Non-covalent thrombin inhibitors featuring P3-heterocycles with P1-bicyclic arginine surrogates
関連化学物質
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3-(acetoxymethyl)-6-methyl-N-(acetyl)aniline
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Peptido sulfonyl fluorides as new powerful proteasome inhibitors
関連化学物質
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C20H25FN4O4S
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Reinventing Hsp90 Inhibitors: Blocking C-Terminal Binding Events to Hsp90 by Using Dimerized Inhibitors
関連化学物質
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macrocycle (Boc)Lys-NMe-D-Phe-Phe-(Cbz)Lys-Leu
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Design, synthesis and structure-activity relationships of 3,5-diaryl-1H-pyrazoles as inhibitors of arylamine N-acetyltransferase
関連化学物質
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5-(3-methoxyphenyl)-3-(4-methoxyphenyl)-1H-pyrazole
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Tuning the moenomycin pharmacophore to enable discovery of bacterial cell wall synthesis inhibitors
関連化学物質
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phenyl 3,4,6-tri-O-acetyl-2-deoxy-1-thio-2-(2,2,2-trichloroethoxycarbonylamino)-β-D-glucopyranoside S-oxide
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N1-alkyl-substituted derivatives of chlorpropamide as inhibitors of aldehyde dehydrogenase.
関連化学物質
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Benzenesulfonamide, 4-chloro-N-[[(1,1-dimethylethyl)amino]carbonyl]-N-ethyl-
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Synthesis of 1-(d-glucopyranosyl)-1,2,3-triazoles and their evaluation as glycogen phosphorylase inhibitors
関連化学物質
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[1-(3',4',5',7'-tetra-O-benzoyl-β-D-gluco-hept-2-ulopyranosyl)-4-phenyl-1,2,3-triazole]onamide
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Toward optimization of the second aryl substructure common to transthyretin amyloidogenesis inhibitors using biochemical and structural studies
関連化学物質
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N-(3,5-dibromo-4-hydroxyphenyl)-2,6-dimethylbenzamide
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Trisubstituted imidazoles as mycobacterium tuberculosis glutamine synthetase inhibitors
関連化学物質
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2-ETHYNYL-6-METHOXYNAPHTHALENE 97
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Discovery of a series of 5-phenyl-2-furan derivatives containing 1,3-thiazole moiety as potent Escherichia coli β-glucuronidase inhibitors
関連化学物質
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5-(4-FLUOROPHENYL)FURAN-2-CARBONYL CHLORIDE
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Aza-Peptide Michael Acceptors: A New Class of Inhibitors Specific for Caspases and Other Clan CD Cysteine Proteases
関連化学物質
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L-Threonine, N-[(phenylmethoxy)carbonyl]-L-leucyl-L-a-glutamyl-, 2-(1,1-dimethylethyl) ester, 3-[2-[2-(1,1-dimethylethoxy)-2-oxoethyl]hydrazide]
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Novel 5α-reductase inhibitors. Synthesis and structure-activity studies of 5-substituted 1-methyl-2-pyridones and 1-methyl-2-piperidones
関連化学物質
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(E)-N,N-diisopropyl-4-<2-(1,2-dihydro-1-methyl-2-oxopyridine-5-yl)ethenyl>benzamide
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Pseudodipeptide Inhibitors of Protein Farnesyltransferase
関連化学物質
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{(R)-1-[((S)-1-Benzylcarbamoyl-propylamino)-methyl]-2-tritylsulfanyl-ethyl}-carbamic acid tert-butyl ester
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1-Aryl-3,4-dihydroisoquinoline inhibitors of JNK3
関連化学物質
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C16H13Cl2NO
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Benzo[c]quinolizin-3-ones: A novel class of potent and selective nonsteroidal inhibitors of human steroid 5α-reductase 1
関連化学物質
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N-BOC-3,4-Dihydro-2(1H)-quinolinone
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Discovery of orally active carboxylic acid derivatives of 2-phenyl-5-trifluoromethyloxazole-4-carboxamide as potent diacylglycerol acyltransferase-1 inhibitors for the potential treatment of obesity and diabetes
関連化学物質
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4-(4-{4-[(2-phenyl-5-trifluoromethyloxazole-4-carbonyl)amino]phenyl}piperazine-1-carbonyl)-trans-cyclohexanecarboxylic acid
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Synthesis and biochemical evaluation of thiochromanone thiosemicarbazone analogues as inhibitors of cathepsin L
関連化学物質
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3-((4-ethylphenyl)thio)propanoic acid
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Targeting the Warburg Effect in cancer; Relationships for 2-arylpyridazinones as inhibitors of the key glycolytic enzyme 6-phosphofructo-2-kinase/2,6-bisphosphatase 3 (PFKFB3)
関連化学物質
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4-(4,5-dibromo-6-oxopyridazin-1(6H)-yl)benzonitrile
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Phenylimidazoles as potent and selective inhibitors of coagulation factor XIa with in vivo antithrombotic activity
関連化学物質
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(S)-2-(2-phenyl-1-(5-phenyloxazol-2-yl)ethyl)isoindoline-1,3-dione
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Discovery of pyrrolidine-2,3-diones as novel inhibitors of p. Aeruginosa pbp3
関連化学物質
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[1-(4-Chloro-phenyl)-meth-(E)-ylidene]-[2-(1H-indol-3-yl)-ethyl]-amine
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Discovery of dihydroisoquinolinone derivatives as novel inhibitors of the p53-MDM2 interaction with a distinct binding mode
関連化学物質
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[4-((R)-sec-Butoxy)-3-methoxy-phenyl]-acetic acid
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Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors
関連化学物質
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trans-1,2-シクロプロパンジカルボン酸
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Novel N-Substituted oseltamivir derivatives as potent influenza neuraminidase inhibitors: Design, synthesis, biological evaluation, ADME prediction and molecular docking studies
関連化学物質
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methyl 4-(3,4-difluorophenyl)-2,4-dioxobutanoate
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SYNTHESIS AND BIOLOGICAL ACTIVITIES OF NEW HMG-COA SYNTHASE INHIBITORS: 2-OXETANONES WITH A SIDE CHAIN CONTAINING BIPHENYL, TERPHENYL OR PHENYLPYRIDINE
関連化学物質
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2-(3-Methylphenyl)isonicotinic acid
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Syntheses of 4-(indole-3-yl)quinazolines - A new class of epidermal growth factor receptor tyrosine kinase inhibitors
関連化学物質
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6-fluoro-5-methylindole-2-carboxylic acid
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N,N′-bisbenzylidenebenzene-1,4-diamines and N,N′- bisbenzylidenenaphthalene-1,4-diamines as sirtuin type 2 (SIRT2) inhibitors
関連化学物質
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Phenol, 4,4'-[1,4-phenylenebis(iminomethylene)]bis-
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6-Phenyl-1H-imidazo[4,5-c]pyridine-4-carbonitrile as cathepsin S inhibitors
関連化学物質
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6-[4-(3-hydroxypropoxy)-3-(trifluoromethyl)-phenyl]-1-methyl-1H-imidazo[4,5-c]pyridine-4-carbonitrile
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Novel quinolizidine salicylamide influenza fusion inhibitors
関連化学物質
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2,5-bis(acetyloxy)benzoic acid
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Improved Inhibitors of Trypanothione Reductase by Combination of Motifs: Synthesis, Inhibitory Potency, Binding Mode, and Antiprotozoal Activities
関連化学物質
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1-((2-(2,6-bis(phenylthio)phenyl)-1H-imidazol-5-yl)methyl)-4-methylpiperazine
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Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors
関連化学物質
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3-(3-PHENOXY-PHENYL)-PROPAN-1-OL
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Modified malto-oligosaccharides as inhibitors of human alpha-amylases
関連化学物質
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p-nitrophenyl-α-D-glucopyranosyl-(1→4)-O-α-D-glucopyranoside
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