ハイスループットスクリーニング
高スループットスクリーニング方法を使用して、ライブラリー中の化合物がAVPによって引き起こされる血管収縮を拮抗する能力を有するかどうかを試験する。これは潜在的な先導化合物を識別するのに役立つだろう。
化学原料を購入する必要がある場合は、 要求情報を送信してください最新の見積りを入手してください。
ハイスループットスクリーニングの学術論文
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Design of potent and selective antagonists of the vasopressor responses to arginine-vasopressin
関連化学物質
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3-MERCAPTO-3-METHYL-BUTYRYL-TYR-PHE-VAL-ASN-CYS-PRO-D-ARG-GLY-NH2
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Synthesis of 4-alkyl-, 4-aryl- and 4-arylamino-5-aminoisoquinolin-1-ones and identification of a new PARP-2 selective inhibitor
関連化学物質
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1-methoxy-5-nitro-4-phenylisoquinoline
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Discovery of an in vivo chemical probe of the lysine methyltransferases G9a and GLP
関連化学物質
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Methyl 5-Methoxy-2-nitro-4-(3-(pyrrolidin-1-yl)propoxy)benzoate
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Screening of a library of hemisalen ligands in asymmetric H-transfer: Reduction of aromatic ketones in water
関連化学物質
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(2,6-dibromo-4-methoxyphenoxy)dimethylphenylsilane
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Improved, selective, human intestinal carboxylesterase inhibitors designed to modulate 7-ethyl-10-[4-(1-piperidino)-1-piperidino]carbonyloxycamptothecin (irinotecan; CPT-11) toxicity
関連化学物質
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ピリジン
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N,N'-(1,4-phenylene)bis(2-fluorobenzenesulfonamide)
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Discovery of Novel and Potent Stearoyl Coenzyme A Desaturase 1 (SCD1) Inhibitors as Anticancer Agents
関連化学物質
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3-Pyridazinecarbonyl chloride, 1,6-dihydro-6-oxo- (9CI)
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Isoxazolopyrimidines as novel F508-CFTR correctors
関連化学物質
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4-isoxazolecarboxamide, 5-amino-3-(3-chlorophenyl)-
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Design, synthesis, and structure-activity relationships of novel insulin receptor tyrosine kinase activators
関連化学物質
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ピリジン
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2-クロロ-5-アミノ安息香酸
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酢酸エチル
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Development of dimeric modulators for anti-apoptotic Bcl-2 proteins
関連化学物質
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C26H24N2O6S4
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Diversity-oriented enantioselective synthesis of highly functionalized cyclic and bicyclic alcohols
関連化学物質
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(-)-(S)-3-vinylcyclohex-2-en-1-yl benzoate
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Achiral oligoamines as versatile tool for the development of aspartic protease inhibitors
関連化学物質
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bis[3-(benzenesulfonylamino)propyl]carbamic acid tert-butyl ester
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Diversity-oriented synthesis-facilitated medicinal chemistry: Toward the development of novel antimalarial agents
関連化学物質
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4-fluoro-N-(((7R,8R,14S)-5-((2S)-1-((4-methoxybenzyl)oxy)propan-2-yl)-1,7,14-trimethyl-4-oxo-4,5,6,7,8,10,11,12,13,14-decahydro-1H-pyrazolo[3,4-b][1,9,5]dioxaazacyclotetradecin-8-yl)methyl)-N-methylbenzenesulfonamide
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Discovery of 2,5-diarylnicotinamides as selective orexin-2 receptor antagonists (2-SORAs)
関連化学物質
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5-(3,5-dichlorophenyl)-N-(3,4-dimethoxybenzyl)-2,3'-bipyridine-3-carboxamide
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A novel route to synthesize libraries of quinoxalines via Petasis methodology in two synthetic operations
関連化学物質
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2-(2-methoxyphenyl)-3-phenylquinoxaline
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Diversity oriented microwave-assisted synthesis of (-)-steganacin aza-analogues
関連化学物質
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butyl-{1-[2'-(tert-butyldimethylsilanyloxymethyl)-4',5'-dimethoxybiphenyl-2-yl]-3-phenylprop-2-ynyl}-amine
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Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors
関連化学物質
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3-(3-PHENOXY-PHENYL)-PROPAN-1-OL
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Reaction discovery by using a sandwich immunoassay
関連化学物質
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2-(4-((tert-butyldimethylsilyl)oxy)-3-methoxyphenyl)acetic acid
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Optimization of 5-phenyl-3-pyridinecarbonitriles as PKCθ inhibitors
関連化学物質
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Nicotinonitrile, 1,4-dihydro-4-oxo- (6CI)
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Benzylidene ketal derivatives as M2 muscarinic receptor antagonists
関連化学物質
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4-[4-(4-methoxy-benzenesulfonyl)-benzoyl]-[1,4']bipiperidinyl-1'-carboxylic acid ethyl ester
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Development of Small Molecules with a Noncanonical Binding Mode to HIV-1 Trans Activation Response (TAR) RNA
関連化学物質
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3-amino-6-methyl-N-(3-(trifluoromethyl)phenyl)thieno[2,3-b]pyridine-2-carboxamide
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Identification of nonpeptidic small-molecule inhibitors of interleukin-2
関連化学物質
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(3-{4-[5-(2,3-dichloro-phenyl)-2-methyl-2H-pyrazol-3-yl]-piperidine-1-sulfonylamino}-propyl)-carbamic acid tert-butyl ester
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Structure-cytotoxicity relationship of a novel series of miconazole-like compounds
関連化学物質
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N-[2-(1H-imidazol-1-yl)-1-phenylethylidene]-N'-phenylhydrazine
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Pyrido<2,1-b>quinazolinecarboxamide Derivatives as Platelet Activating Factor Antagonists
関連化学物質
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(R)-2-AMINO-5-(3-PYRIDYL)PENTANE
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New oxadiazolidinedione derivatives as potent and selective human β3 agonists
関連化学物質
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tert-butyl 2-{2,4-dioxo-5-[4-(4-oxo-1-piperidinyl)benzyl]-1,3-thiazolidin-3-yl}acetate
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Discovery of 8-Amino-imidazo[1,5-a]pyrazines as Reversible BTK Inhibitors for the Treatment of Rheumatoid Arthritis
関連化学物質
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4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-N-(4-trifluoromethyl-pyridin-2-yl)benzamide
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Approaches to the high-throughput synthesis of analogues of dihydroaertiginoic acid
関連化学物質
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L-Cysteine, N-(2-hydroxybenzoyl)-
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Structure-activity relationships of diphenylpiperazine N-type calcium channel inhibitors
関連化学物質
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1-(o-Chloro-α-phenylbenzyl)piperazine
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Parallel solid-phase synthesis of zatebradine analogues as potential If channel blockers
関連化学物質
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7,8-Dimethoxy-3-(3-iodopropyl)-1,3-dihydro-2H-3-benzazepin-2-one
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Isoxazole carboxylic acids as protein tyrosine phosphatase 1B (PTP1B) inhibitors
関連化学物質
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3-Isoxazolecarboxylic acid, 4-amino-5-[3-[(1E)-3-hydroxy-1-propenyl]phenyl]-, ethyl ester
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Small-molecular, non-peptide, non-ATP-competitive polo-like kinase 1 (Plk1) inhibitors with a terphenyl skeleton
関連化学物質
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3,5-Difluoro-4-hydroxybenzeneboronic acid pinacol ester, 96%
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α-Hydroxy Phosphinyl-Based Inhibitors of Human Renin
関連化学物質
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N-[(2S)-2-{[1-(cyclohexylmethyl)-2-(dimethoxyphosphoryl)-2-hydroxyethyl]amino}-4-methylpentanoyl]-Nalpha-(cyclopentylcarbonyl)-L-phenylalaninamide
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Selective inhibition of type II dehydroquinases
関連化学物質
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3-deoxyquinic acid
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8-Substituted 3,4-dihydroquinolinones as a novel scaffold for atypical antipsychotic activity
関連化学物質
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Benzoylcholine Chloride
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2,5,6-Trisubstituted imidazo[2,1-b][1,3,4]thiadiazoles: Search for antihyperlipidemic agents
関連化学物質
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N-((2-(benzo[d][1,3]dioxol-5-yl)-6-phenylimidazo[2,1-b][1,3,4]thiadiazol-5-yl)methylene)aniline
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Discovery of the First Environment-Sensitive Fluorescent Probe for GPR120 (FFA4) Imaging
関連化学物質
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methyl 4-[(4-nitrophenyl)methoxy]benzenepropanoate
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Discovery of novel urea-based hepatitis C protease inhibitors with high potency against protease-inhibitor-resistant mutants
関連化学物質
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N-(6-acetyl-3-methoxy-2-methylphenyl)-4-cyclopropylthiazole-2-carboxamide
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Structure-Activity Relationships of 9-Alkyladenine and Ribose-Modified Adenosine Derivatives at Rat A3 Adenosine Receptors
関連化学物質
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9H-Purin-6-amine, 2-chloro-N-[(3-iodophenyl)methyl]-9-methyl-
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1H-indole derivatives as calcium antagonists
関連化学物質
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[3-(1-Hydroxy-propyl)-2-methyl-5-nitro-indol-1-yl]-phenyl-methanone
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2-acetylphenol analogs as potent reversible monoamine oxidase inhibitors
関連化学物質
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1-(4-(4-cyanobenzyloxy)-2-hydroxyphenyl)ethanone
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New benzimidazoles as thrombopoietin receptor agonists
関連化学物質
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(E)-3-(4-Acetylamino-3-nitro-phenyl)-2-methyl-acrylic acid ethyl ester
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Identification of Darmstoff analogs as selective agonists and antagonists of lysophosphatidic acid receptors
関連化学物質
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1,3-Dioxolane-4-methanol, 2-(8Z)-8-heptadecenyl-
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