体外評価
合成した化合物のゼラチナーゼに対する阻害活性を体外試験した。酵素分析やゼラチナーゼスペクトルなどの技術はそれらの有効性を評価することができる。ゼラチナーゼ阻害のアナモルの範囲内にあるべきIC 50値を決定する必要があります。
化学原料を購入する必要がある場合は、 要求情報を送信してください最新の見積りを入手してください。
体外評価の学術論文
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Design, Synthesis, and Biological Evaluation of Tetrahydro-β-carboline Derivatives as Selective Sub-Nanomolar Gelatinase Inhibitors
関連化学物質
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(1RS)-2-(4''-methoxy-4'-phenoxybenzenesulfonyl)-1,2,3,4-tetrahydro-norarmano-1-carboxylic acid
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Design, synthesis, and biological evaluation of new raloxifene analogues of improved antagonist activity and endometrial safety
関連化学物質
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(4-(2-hydroxyethoxy)phenyl)(6-methoxy-2-(4-methoxyphenyl)benzo[b]thiophen-3-yl)methanone
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Synthesis and evaluation of β-carboline derivatives as potential monoamine oxidase inhibitors
関連化学物質
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7-(phenethoxy)-1-methyl-β-carboline
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Design, synthesis, and in vitro evaluation of aza-peptide aldehydes and ketones as novel and selective protease inhibitors
関連化学物質
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L-Alanine, N-[(phenylmethoxy)carbonyl]-L-alanyl-, hydrazide
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Towards to hENT1-nucleoside transporter selective imaging agents. Synthesis and in vitro evaluation of the radiolabeled SAENTA analogues
関連化学物質
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12,13-Dithia-2,9,16,23-tetraazatetracosanedioic acid, 8,17-dioxo-, bis(1,1-dimethylethyl) ester
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Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) Family
関連化学物質
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Propanedioic acid, methyl-, monoethyl ester, potassium salt
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Synthesis and in vitro evaluation of tetrahydroisoquinolinyl benzamides as ligands for σ receptors
関連化学物質
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4-(3,4-dimethoxyphenethylamino)butanenitrile
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Synthesis, in vitro, and in vivo evaluation of phosphate ester derivatives of combretastatin A-4
関連化学物質
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diisopropyl-phosphoramidous acid 2-cyano-ethyl ester cyclohexyl ester
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Synthesis and in vitro evaluation of xylene linked carbamoyl bis-pyridinium monooximes as reactivators of organophosphorus (OP) inhibited electric eel acetylcholinesterase (AChE)
関連化学物質
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1-(2-bromomethylbenzyl)-3-hydroxyiminomethylpyridinium bromide
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Synthesis, in vitro and in vivo evaluation of novel substituted N-(4-(2-(4-benzylpiperazin-1-yl)ethoxy)phenyl)-N-methyl-quinazolin-4-amines as potent antitumor agents
関連化学物質
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1-(2-Chloroethyl)-4-[(2-fluorophenyl)methyl]piperazine
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New fluorinated dopamine D2 ligands with benzofuran skeleton. The synthesis and in vitro evaluation
関連化学物質
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7-carboxy-5-ethyl-2,3-dihydrobenzofuran
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